Aminoborylation/Suzuki-Miyaura tandem cross coupling of aryl iodides as efficient and selective synthesis of unsymmetrical biaryls.

نویسندگان

  • Ludovic Marciasini
  • Nicolas Richy
  • Michel Vaultier
  • Mathieu Pucheault
چکیده

Sequential borylation of a first aryl iodide using a dialkylaminoborane followed by a Suzuki-Miyaura cross coupling of second aryl iodide ended up with an efficient, selective and practical synthesis of unsymmetrical biaryls. This tandem coupling shows a wide range of applicability.

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عنوان ژورنال:
  • Chemical communications

دوره 48 10  شماره 

صفحات  -

تاریخ انتشار 2012